BQ-3020 TFA (143113-45-5 free base)
CAS No. ——
BQ-3020 TFA (143113-45-5 free base)( —— )
Catalog No. M30404 CAS No. ——
BQ-3020 (TFA) is a selective ETB receptor agonist that inhibits [125I] et-1 binding to the ETB receptor in the cerebellum with a 0.2nm IC50, causing vasoconstriction.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameBQ-3020 TFA (143113-45-5 free base)
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NoteResearch use only, not for human use.
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Brief DescriptionBQ-3020 (TFA) is a selective ETB receptor agonist that inhibits [125I] et-1 binding to the ETB receptor in the cerebellum with a 0.2nm IC50, causing vasoconstriction.
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DescriptionBQ-3020 (TFA) is a selective ETB receptor agonist that inhibits [125I] et-1 binding to the ETB receptor in the cerebellum with a 0.2nm IC50, causing vasoconstriction.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorIC50: 0.2 nM ([125I]ET-1 binding to ETB receptor)
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight2120.35
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Molecular FormulaC98H141F3N20O27S
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical NameSequence:N-Acetyl-Leu-Met-Asp-Lys-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu-Asp-Ile-Ile-Trp
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
Ihara M, et al. A novel radioligand [125I]BQ-3020 selective for endothelin (ETB) receptors. Life Sci. 1992;51(6):PL47-52.
molnova catalog
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